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Brand Model and Executive

Management Case No 4. NSAIDS.

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Indomethacin āĻĄā§āϰāĻžāĻ— āĻ…āĻĢ āϚāϝāĻŧ⧇āϜ for- Gout, Ankylosing Spondylitis , Musculoskeletal pain__

Capsule1. Indomet SR 75mg (AS A Indomethacin Drugs for Osteoarthritis, Drugs used for Rheumatoid Arthritis, Non-steroidal Anti-inflammatory Drugs (NSAIDs).

Paracetamol Safest in āĻĒā§āϰ⧇āĻ—āĻ¨ā§āϝāĻžāĻ¨ā§āϏāĻŋ Analgesic āĻāϰ āϜāĻ¨ā§āϝ

Ketorolac āϚāϝāĻŧ⧇āϜ āĻ…āĻĢ āĻĄā§āϰāĻžāĻ— Mild to Moderate Post operative Pain**Also Diclofenac_

Tablet 1.Torax 10mg (AS A Ketorolac Tromethamine Drugs used for Rheumatoid Arthritis, Non-Opioid Analgesics).

Dysmenorrhea āϤ⧇ āϚāϝāĻŧ⧇āϜ Mefenamic Acid**

Tablet 1:-Myfocin 500 mg AS A Mefenamic Acid As a Drugs for Osteoarthritis, Drugs used for Rheumatoid Arthritis, Non-steroidal Anti-inflammatory Drugs (NSAIDs)

Most Hepatotoxic – Sulindac & Diclofenac

Tablet 1:-Sulidac 200mg AS A Sulindac Drugs for Osteoarthritis, Drugs used for Rheumatoid Arthritis, Drugs used in Gout, Non-steroidal Anti-inflammatory Drugs (NSAIDs).

Tablet 2:-Clofenac SR 100mg AS A Diclofenac Sodium Drugs for Osteoarthritis, Drugs used for Rheumatoid Arthritis, Non-steroidal Anti-inflammatory Drugs (NSAIDs).

Most Nephrotoxic- Ketorolac & Indomethacin*

Safest NSAIDs in Cardiac pt -Naproxen

Tablet 1.Naproxen 500mg AS A Naproxen Sodium AS A Drugs for Osteoarthritis, Drugs used for Rheumatoid Arthritis, Non-steroidal Anti-inflammatory Drugs (NSAIDs).

Safest NSAIDs in PUD – Ibuprofen Etorix/tory 60 mg.

Highest efficacy NSAID is – Diclofenac 150 mg/day

Tablet 2:-Clofenac SR 100mg AS A Diclofenac Sodium Drugs for Osteoarthritis, Drugs used for Rheumatoid Arthritis, Non-steroidal Anti-inflammatory Drugs (NSAIDs).

Safest NSAIDs in Renal Failure – Sulindac,and Nabumetone

Tablet 1:-Sulidac 200mg AS A Sulindac Drugs for Osteoarthritis, Drugs used for Rheumatoid Arthritis, Drugs used in Gout, Non-steroidal Anti-inflammatory Drugs (NSAIDs).

Tablet 2.Buflex 500mg (AS A Nabumetone AS A Drugs for Osteoarthritis, Drugs used for Rheumatoid Arthritis).

Safest NSAIDs in IHD/Heart Failure – Aspirin

āĻāĻ•āϏāĻžāĻĨ⧇ 1 āĻāϰ āĻŦ⧇āĻļāĻŋ NSAID & Long term āχāωāϏ āĻ•āϰāϞ⧇ Analgesic Nephropathy āĻšāϤ⧇ āĻĒāĻžāϰ⧇

NSAID induced PUD āϤ⧇ Co prescription āĻšāĻŋāϏ⧇āĻŦ⧇ PPi / Misoprostol

Tablet 1:-Cytomis As a Misoprostol (As a Drugs acting on the Uterus, Prostaglandin analogues).

Immediate After āĻŦāĻžāĻ°ā§āύ (after burn there may B Curling ulcer) So avoid NSAID

āĻŦāĻžāĻšā§āϚāĻžāĻĻ⧇āϰ āĻ­āĻžāχāϰāĻžāϞ āχāύāĻĢ⧇āĻ•āĻļāύ āĻ (Influenza B & Chikn pox) Avoid Aspirin To reduce Fever**(Reye’s Syndrome )āĻšāϤ⧇ āĻĒāĻžāϰ⧇

Paracetamol maximum āĻĄā§‹āϏ āĻĄā§‡āχāϞāĻŋ āύāϰāĻŽāĻžāϞ person āĻāϰ āĻ•ā§āώ⧇āĻ¤ā§āϰ⧇ 4 gm

Paracetamol āĻĒāϝāĻŧāϏāύāĻŋāĻ‚ Antidote-(N Acetylcystine )

COX -2 āĻšāϞ⧋ Strongest NSAID & āĻāϰ GIT Side effects āĻ•āĻŽ..GI irritation āĻ•āϰ⧇ āύāĻž,, Avoid in (IHD & āĻŦāϝāĻŧāĻ¸ā§āĻ• āĻĒ⧇āĻļ⧇āĻ¨ā§āϟ )

Tablet 1:-Tory 120 mg AS A Etoricoxib AS A Non-steroidal Anti-inflammatory Drugs (NSAIDs).

āĻŦāĻžāĻšā§āϚāĻžāĻĻ⧇āϰ āϜāĻ¨ā§āϝ āĻŦ⧇āĻ¸ā§āϟ āϚāϝāĻŧ⧇āϜ Paracetamol thn Ibuprofen

Salfasalazine āĻĒā§āϰ⧇āĻ—āĻ¨ā§āϝāĻžāĻ¨ā§āϏāĻŋāϤ⧇ use āĻ•āϰāĻž āϝ⧇āϤ⧇ āĻĒāĻžāϰ⧇ āĻ•āĻŋāĻ¨ā§āϤ⧁ Breastfeeding āĻ Contraindicated

Tablet 1.Salazine 500mg AS A Salfasalazine AS A Drugs for Irritable Bowel Syndrome, Drugs used for Rheumatoid Arthritis, Ulcerative Colitis.

Chronic use of NSAID – āϕ⧋āϞāύ Cancer āĻāϰ āϰāĻŋāĻ¸ā§āĻ• āĻ•āĻŽāĻžāϝāĻŧ

Raiyyan Tahsan Date:-27-12-2024 Friday Time:-7-21-30 PM.

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